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Enade Perdana Istyastono
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Year
Synthesis and QSAR of Quinazoline Sulfonamides As Highly Potent Human Histamine H4 Receptor Inverse Agonists
RA Smits, M Adami, EP Istyastono, OP Zuiderveld, CME van Dam, ...
Journal of medicinal chemistry 53 (6), 2390-2400, 2010
1352010
Molecular determinants of ligand binding to H4R species variants
HD Lim, C de Graaf, W Jiang, P Sadek, PM McGovern, EP Istyastono, ...
Molecular pharmacology 77 (5), 734-743, 2010
792010
Virtual Fragment Screening: Discovery of Histamine H3 Receptor Ligands Using Ligand-Based and Protein-Based Molecular Fingerprints
F Sirci, EP Istyastono, HF Vischer, AJ Kooistra, S Nijmeijer, M Kuijer, ...
Journal of chemical information and modeling 52 (12), 3308-3324, 2012
782012
PyPLIF: Python-based Protein-Ligand Interaction Fingerprinting
M Radifar, N Yuniarti, EP Istyastono
Bioinformation 9 (6), 325-328, 2013
772013
Molecular Determinants of Ligand Binding Modes in the Histamine H4 Receptor: Linking Ligand-Based Three-Dimensional Quantitative Structure–Activity …
EP Istyastono, S Nijmeijer, HD Lim, A van de Stolpe, L Roumen, ...
Journal of medicinal chemistry 54 (23), 8136-8147, 2011
662011
Triazole Ligands Reveal Distinct Molecular Features That Induce Histamine H4 Receptor Affinity and Subtly Govern H4/H3 Subtype Selectivity
M Wijtmans, C de Graaf, G de Kloe, EP Istyastono, J Smit, H Lim, ...
Journal of medicinal chemistry 54 (6), 1693-1703, 2011
502011
Clobenpropit analogs as dual activity ligands for the histamine H3 and H4 receptors: synthesis, pharmacological evaluation, and cross-target QSAR studies
HD Lim, EP Istyastono, A van de Stolpe, G Romeo, S Gobbi, M Schepers, ...
Bioorganic & medicinal chemistry 17 (11), 3987-3994, 2009
422009
Structure-based virtual screening for fragment-like ligands of the G protein-coupled histamine H 4 receptor
EP Istyastono, AJ Kooistra, HF Vischer, M Kuijer, L Roumen, S Nijmeijer, ...
MedChemComm 6 (6), 1003-1017, 2015
412015
Matrix metalloproteinase 9 (MMP9) in wound healing of diabetic foot ulcer: Molecular target and structure-based drug design
M Hariono, SH Yuliani, EP Istyastono, FDO Riswanto, CF Adhipandito
Wound Medicine 22, 1-13, 2018
362018
Structure-based design of eugenol analogs as potential estrogen receptor antagonists
Y Anita, M Radifar, LBS Kardono, M Hanafi, EP Istyastono
Bioinformation 8 (19), 901, 2012
362012
Molecular determinants of selective agonist and antagonist binding to the histamine H4 receptor
E P Istyastono, C de Graaf, I JP de Esch, R Leurs
Current Topics in Medicinal Chemistry 11 (6), 661-679, 2011
362011
Inhibition of human glutathione S-transferases by curcumin and analogues
R Appiah-Opong, JNM Commandeur, E Istyastono, JJ Bogaards, ...
Xenobiotica 39 (4), 302-311, 2009
362009
Natural peptides in drug discovery targeting acetylcholinesterase
V Prasasty, M Radifar, E Istyastono
Molecules 23 (9), 2344, 2018
342018
Employing recursive partition and regression tree method to increase the quality of structure-based virtual screening in the estrogen receptor alpha ligands identification
EP Istyastono
Asian J. Pharm. Clin. Res 8 (6), 21-24, 2015
242015
The cytotoxic activity on T47D breast cancer cell of genistein-standardized ethanolic extract of tempeh-A fermented product of soybean (Glycine max)
SH Yuliani, EP Istyastono, FDO Riswanto
Orient. J. Chem 32 (3), 1619-1624, 2016
222016
PyPLIF-assisted redocking indomethacin-(R)-alpha-ethyl-ethanolamide into cyclooxygenase-1
M Radifar, N Yuniarti, EP Istyastono
Indonesian Journal of Chemistry 13 (3), 283-286, 2013
212013
The importance of ARG513 as a hydrogen bond anchor to discover COX-2 inhibitors in a virtual screening campaign.
N Yuniarti, Z Ikawati, EP Istyastono
Bioinformation 6 (4), 164-166, 2011
202011
Retrospective validation of a structure-based virtual screening protocol to identify ligands for estrogen receptor alpha and its application to identify the alpha-mangostin …
A Setiawati, FDO Riswanto, SH Yuliani, EP Istyastono
Indonesian Journal of Chemistry 14 (2), 103-108, 2014
192014
Perbandingan stabilitas fisis sediaan nanoemulsi minyak biji delima dengan fase minyak long-chain triglyceride dan medium-chain triglyceride
SH Yuliani, M Hartini, BP Stephanie, EP Istyastono
Traditional Medicine Journal 21 (2), 94, 2016
172016
Binary quantitative structure-activity relationship analysis in retrospective structure based virtual screening campaigns targeting estrogen receptor alpha
EP Istyastono, N Yuniarti, M Hariono, SH Yuliani, FDO Riswanto
Asian J. Pharm. Clin. Res 10 (12), 206-211, 2017
162017
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