| Synthesis and biological evaluation of spiro [cyclopropane-1, 3′-indolin]-2′-ones as potential anticancer agents CN Reddy, VL Nayak, GS Mani, JS Kapure, PR Adiyala, RA Maurya, ... Bioorganic & Medicinal Chemistry Letters 25 (20), 4580-4586, 2015 | 75 | 2015 |
| Visible-light photoredox catalysis: direct synthesis of fused β-carbolines through an oxidation/[3+ 2] cycloaddition/oxidative aromatization reaction cascade in batch and flow … D Chandrasekhar, S Borra, JS Kapure, GS Shivaji, G Srinivasulu, ... Organic Chemistry Frontiers 2 (10), 1308-1312, 2015 | 59 | 2015 |
| Synthesis of phenstatin/isocombretastatin–chalcone conjugates as potent tubulin polymerization inhibitors and mitochondrial apoptotic inducers A Kamal, GB Kumar, M Vishnuvardhan, AB Shaik, VS Reddy, R Mahesh, ... Organic & biomolecular chemistry 13 (13), 3963-3981, 2015 | 53 | 2015 |
| Combretastatin linked 1, 3, 4-oxadiazole conjugates as a Potent Tubulin Polymerization inhibitors A Kamal, PS Srikanth, M Vishnuvardhan, GB Kumar, KS Babu, ... Bioorganic Chemistry 65, 126-136, 2016 | 49 | 2016 |
| Rapid access to novel 1, 2, 3-triazolo-heterocyclic scaffolds via tandem knoevenagel condensation/azide–alkyne 1, 3-dipolar cycloaddition reaction in one pot RA Maurya, PR Adiyala, D Chandrasekhar, CN Reddy, JS Kapure, ... ACS Combinatorial Science 16 (9), 466-477, 2014 | 42 | 2014 |
| Discovery of pyrrolospirooxindole derivatives as novel cyclin dependent kinase 4 (CDK4) inhibitors by catalyst-free, green approach A Kamal, R Mahesh, VL Nayak, KS Babu, GB Kumar, AB Shaik, ... European Journal of Medicinal Chemistry 108, 476-485, 2016 | 37 | 2016 |
| Synthesis and biological evaluation of 1, 2, 3-triazole linked aminocombretastatin conjugates as mitochondrial mediated apoptosis inducers A Kamal, B Shaik, VL Nayak, B Nagaraju, JS Kapure, MS Malik, TB Shaik, ... Bioorganic & medicinal chemistry 22 (19), 5155-5167, 2014 | 35 | 2014 |
| Diastereoselective synthesis of spiro [cyclopropane-1, 3′-indolin]-2′-ones through metal-free cyclopropanation using tosylhydrazone salts JS Kapure, CN Reddy, PR Adiyala, R Nayak, VL Nayak, JB Nanubolu, ... RSC advances 4 (72), 38425-38432, 2014 | 34 | 2014 |
| A New Selective Pharmacological Enhancer of the Orai1 Ca2+ Channel Reveals Roles for Orai1 in Smooth and Skeletal Muscle Functions I Azimi, RJ Stevenson, X Zhang, A Meizoso-Huesca, P Xin, M Johnson, ... ACS pharmacology & translational science 3 (1), 135-147, 2020 | 30 | 2020 |
| Catalyst-free stereoselective cyclopropanation of electron deficient alkenes with ethyl diazoacetate RA Maurya, JS Kapure, PR Adiyala, PS Srikanth, D Chandrasekhar, ... RSC Advances 3 (36), 15600-15603, 2013 | 28 | 2013 |
| Synthesis of α-amino amidines through molecular iodine-catalyzed three-component coupling of isocyanides, aldehydes and amines PR Adiyala, D Chandrasekhar, JS Kapure, CN Reddy, RA Maurya Beilstein Journal of Organic Chemistry 10 (1), 2065-2070, 2014 | 27 | 2014 |
| Design and synthesis of 1, 2, 3-triazolo linked benzo [d] imidazo [2, 1-b] thiazole conjugates as tubulin polymerization inhibitors SP Shaik, M Vishnuvardhan, F Sultana, AVS Rao, C Bagul, ... Bioorganic & Medicinal Chemistry 25 (13), 3285-3297, 2017 | 25 | 2017 |
| Synthesis and biological evaluation of benzimidazole–oxindole conjugates as microtubule-targeting agents A Kamal, B Nagaseshadri, VL Nayak, V Srinivasulu, M Sathish, JS Kapure, ... Bioorganic chemistry 63, 72-84, 2015 | 25 | 2015 |
| Synthesis and biological evaluation of arylcinnamide linked combretastatin-A4 hybrids as tubulin polymerization inhibitors and apoptosis inducing agents A Kamal, S Bajee, VL Nayak, AVS Rao, B Nagaraju, CR Reddy, ... Bioorganic & Medicinal Chemistry Letters 26 (12), 2957-2964, 2016 | 24 | 2016 |
| Highly diastereoselective synthesis of spiro [cyclopropane-1, 3′-indolin]-2′-ones via catalyst-free cyclopropanation using ethyl diazoacetate RA Maurya, CN Reddy, GS Mani, JS Kapure, PR Adiyala, JB Nanubolu, ... Tetrahedron 70 (32), 4709-4717, 2014 | 24 | 2014 |
| Regio-and stereoselective synthesis of novel spiropyrrolidines through 1, 3-dipolar cycloaddition reactions of azomethine ylides and 2-styrylquinazolin-4 (3 H)-ones RA Maurya, R Nayak, CN Reddy, JS Kapure, JB Nanubolu, KK Singarapu, ... RSC advances 4 (61), 32303-32311, 2014 | 22 | 2014 |
| Design and synthesis of aminostilbene–arylpropenones as tubulin polymerization inhibitors A Kamal, GB Kumar, S Polepalli, AB Shaik, VS Reddy, MK Reddy, ... ChemMedChem 9 (11), 2565-2579, 2014 | 21 | 2014 |
| Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screening JA Miles, JS Kapure, GS Deora, C Courageux, A Igert, J Dias, ... Bioorganic & Medicinal Chemistry Letters 30 (24), 127609, 2020 | 7 | 2020 |
| Small Molecule Anti-Inflammatory TYK2 Inhibitors Attenuate Inflammation and Clinical Symptoms in a Mouse Model of Imiquimod Induced Psoriasis SB Mallik, A Tandon, JA Kuriappan, JS Kapure, M Halle, A Iyer Journal of Pharmacology and Experimental Therapeutics 385 (S3), 2023 | | 2023 |
| Topical selective TYK2 inhibition attenuates inflammation and clinical symptoms in a mouse model of human psoriasis SB Mallik, A Tandon, JA Kuriappan, JS Kapure, M Halle, A Iyer The Journal of Immunology 210 (1_Supplement), 166.05-166.05, 2023 | | 2023 |
Ram Awatar MauryaCSIR-North East Institute of Science & Technology JorhatBestätigte E-Mail-Adresse bei neist.res.in
